CDK Family


Continuous proliferation is an important hallmark of tumor cells, blocking the tumor cell cycle has become an important means to control tumor development. The complex of cyclin and cyclin dependent kinases (CDKs) can control the cell division, and the development of inhibitors around this family has become an important branch of drug development in the field of cancer in recent years.

 

CDKs, belonging to the serine/threonine protein kinase family. CDKs binds to the corresponding regulatory subunit-cyclin to form an active heterodimer, which is mainly involved in cell cycle regulation and transcriptional regulation (Figure 1). CDK1, CDK4, CDK6, etc., involved in the cell cycle include, and CDK7, CDK8, CDK9, etc., involved in transcriptional regulation.

 

Biortus Biortus

 

 

 

The Biortus Protein Catalogue currently offers 33 CDK/cyclin complex proteins (Table 1), with specific in-house biochemical assays for all the proteins readily available. 

 

Catalog No.

Organism

Expression system

Tag

Sequence

CDK1/Cyclin B1-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-M297/N165-V433

CDK1/Cyclin A2-H21A

Homo sapiens

Insect cell

GST/His

M1-M297/E174-L432

CDK1/Cyclin E1-H21A

Homo sapiens

Insect cell

GST/His

M1-M297/M1-E410

CDK1/Cyclin E2-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-M297/S2-H404

CDK2/Cyclin A2-H21A

Homo sapiens

Insect cell

GST/His

M1-L298/E174-L432

CDK2/Cyclin E1-H21A

Homo sapiens

Insect cell

GST/His

M1-L298/M1-E410

CDK2/Cyclin D1-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-L298/M1-I295

CDK2/Cyclin O-H214A

Homo sapiens

Insect cell

GST/His-Flag

M1-L298/V2-S349

CDK2/Cyclin E2-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-L298/S2-H404

CDK3/Cyclin E1-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-H305/M1-E410

CDK4/Cyclin D2-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-E303/E2-L289

CDK6/Cyclin D3-H21A

Homo sapiens

Insect cell

GST/His

M1-A326/M1-L292

CDK6/Cyclin D1-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-A326/M1-I295

CDK6/Cyclin D2-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-A326/E2-L289

CDK7/Cyclin H/MAT1-H211A

Homo sapiens

Insect cell

GST/His/His

M1-F346/M1-L323/M1-S309

CDK8/Cyclin C/MED12-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-Y464/M1-S283/M1-D100

CDK9/Cyclin T1-H21A

Homo sapiens

Insect cell

GST/His

M1-F372/M1-K726

CDK9/Cyclin K-H24A

Homo sapiens

Insect cell

GST/Flag

M1-F372/M1-S300

CDK9/Cyclin T2-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-F372/A2-N663

CDK15/Cyclin Y-H24A

Homo sapiens

Insect cell

GST/Flag

M1-W435/M1-S341

CDK16/Cyclin Y-H24A

Homo sapiens

Insect cell

GST/Flag

M1-F496/M1-S341

CDK19/Cyclin C/MED12-H241A

Homo sapiens

Insect cell

GST/Flag-His

M1-Y502/M1-S283/M1-D100

 

 

See All Recombinant Proteins >>>
For custom CDK/Cyclin generation, please see Protein Generation or contact info@wuxibiortus.com.

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